Words similar to antagonist
Example sentences for: antagonist
How can you use “antagonist” in a sentence? Here are some example sentences to help you improve your vocabulary:
The GABAa antagonist bicuculline also widened vertebral arch distance at the 0.5 and 1 mg/kg doses (p < .05), but not at the 2 mg/kg dose.
These would be drugs that act as an agonist at one receptor and as an antagonist or partial agonist at another receptor type.
Hibert et al proposed an early model for the antagonist pharmacophore of the 5-HT 3 R [ 18 ] . According to this model, all 5-HT 3 R antagonists contain an aromatic ring, a carbonyl oxygen or bioisosteric equivalent, and a basic nitrogen.
While both these ligands bind with high affinities (less than 1 nM) to μ opioid receptors, WIN 44,441 acts as an antagonist at μ opioid receptors and xorphanol is a very weak agonist at μ opioid receptor (Gharagozlou et al.
These results strongly support the model, initially hypothesized for cyclopamine [ 11 ] , that the reduced potency observed for Hh antagonists on Smo act-expressing cells is directly due to a reduced affinity of the antagonist for the mutated Smo protein.
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