Words similar to etorphine
Example sentences for: etorphine
How can you use “etorphine” in a sentence? Here are some example sentences to help you improve your vocabulary:
All ligands were dissolved in distilled water except cyclazocine, dezocine, etorphine, which were dissolved in 100% ethanol.
In a study carried out in vivo on guinea pig ileum ( 18), the authors showed a rapid endocytosis of the μ-opioid receptor in neurons in response to etorphine stimulation but not after morphine administration.
The rank order of efficacy of the ligands tested were fentanyl = hydromorphone = β-endorphin > etorphine = lofentanil = butorphanol = morphine= nalbuphine = nalorphine > cyclazocine = dezocine = metazocine ≥ xorphanol.
The IC 50 of all ligands studied were between 1-10 nM, with the exception of etorphine, which was the most potent drug, with an IC 50 of 0.3 nM, morphine, which was the least potent drug with an IC 50 of 12 nM and the endogenous ligand β-endorphin with IC 50 of 500 nM.
Loading...