Words similar to etorphine
Example sentences for: etorphine
How can you use “etorphine” in a sentence? Here are some example sentences to help you improve your vocabulary:
Based on these analyses, there was no difference in the efficacy of butorphanol, etorphine, lofentanil or nalorphine compared to fentanyl or hydromorphone (p > 0.05).
The rank order of efficacy of the ligands tested was metazocine = xorphanol ≥ fentanyl = SKF 10047 = etorphine = hydromorphone = butorphanol = lofentanil > WIN 44,441 = Nalbuphine = cyclazocine ≥ met-enkephalin >> morphine = dezocine.
The IC 50 of all ligands studied were between 1-10 nM, with the exception of etorphine, which was the most potent drug, with an IC 50 of 0.3 nM, morphine, which was the least potent drug with an IC 50 of 12 nM and the endogenous ligand β-endorphin with IC 50 of 500 nM.
Antagonists were defined as ligands that were able to repeatedly block the inhibitory effect of 1 nM etorphine on forskolin-stimulated cAMP production.
Finally, a dose response curve of naltrexone as it fully blocked the effect of 1 nM etorphine is shown (Fig 1d).