Words similar to cpbg
Example sentences for: cpbg
How can you use “cpbg” in a sentence? Here are some example sentences to help you improve your vocabulary:
In contrast to 5-HT and m CPBG, however, lerisetron also interacts with Y152 as indicated by the 190 fold increase in K i on Y152A mutant receptors.
This difference in binding site interactions of the antagonist d -tc and the agonists 5-HT and m CPBG could be the result of a slightly different positioning of d -tc in the binding site.
al . have suggested that W183 may be involved in a cation-π interaction with the amino group of 5-HT and m CPBG [ 26 ] . If W183 and Y142 are located near each other but on opposite faces of the binding site in the 5-HT 3 R, then they could potentially act in concert to help stabilize a conformation of the receptor leading to channel opening.
This increase in K i indicates an important interaction of lerisetron with Y142 and a similarity between the binding location of lerisetron, 5-HT and m CPBG.
[ 3H]granisetron does not appear to interact with any of the amino acids tested while d -tc interacts with only Y140, m CPBG and 5-HT with Y142 and lerisetron with both Y142 and Y152.
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