Words similar to xorphanol
Example sentences for: xorphanol
How can you use “xorphanol” in a sentence? Here are some example sentences to help you improve your vocabulary:
Clinically, xorphanol is a well tolerated, orally active analgesic that provides effective pain relief but shows low physical dependence liability [ 29 30 ] . It is possible that the low physical dependence liability of this drug is due to its partial agonism at μ opioid receptors.
Moreover, until now the activity of xorphanol at δ opioid receptors had not been described.
The rank order of affinity of the ligands was xorphanol > Win 44,441> nalorphine > morphine ≥ nalbuphine > fentanyl (Table 2).
In fact one of the most potent ligands, xorphanol, was the least efficacious.
The most potent ligands studied, as measured by the lowest IC 50 values (Table 1), were etorphine, cyclazocine, lofentanil, and xorphanol with IC 50 's of less than 10 nM.