Words similar to xorphanol
Example sentences for: xorphanol
How can you use “xorphanol” in a sentence? Here are some example sentences to help you improve your vocabulary:
Moreover, until now the activity of xorphanol at δ opioid receptors had not been described.
Both these ligands have high affinities and potencies at δ opioid receptors with xorphanol being very efficacious at δ opioid receptors.
The most potent ligands studied, as measured by the lowest IC 50 values (Table 1), were etorphine, cyclazocine, lofentanil, and xorphanol with IC 50 's of less than 10 nM.
Clinically, xorphanol is a well tolerated, orally active analgesic that provides effective pain relief but shows low physical dependence liability [ 29 30 ] . It is possible that the low physical dependence liability of this drug is due to its partial agonism at μ opioid receptors.
The rank order of potency of these ligands was; etorphine>lofentanil≥cyclazocine=xorphanol>met-enkephalin> Win 44,441=hydromorphone≥butorphanol>metazocine=SKF 10047> dezocine≥ nalbuphine>morphine>fentanyl.