Words similar to lerisetron
Example sentences for: lerisetron
How can you use “lerisetron” in a sentence? Here are some example sentences to help you improve your vocabulary:
These data support our hypothesis that Y142 interacts with the distal piperazine nitrogen of lerisetron.
The increases in the K i values were 190 fold for lerisetron, 98 fold for analog 1 and only 40 fold for analog 2. Thus, analog 1 retains much of its ability to interact with Y152 despite the absence of the N-benzyl group, while analog 2 interacts more weakly with this amino acid.
Our data does not support an interaction of this amino acid with either the N-benzyl or benzimidazole portions of lerisetron.
A loop structure would bring them into closer proximity and permit interaction with the small molecule lerisetron.
i for analog 2 suggests that analog 2 binds weakly to Y152 while lerisetron and analog 1 bind more tightly.
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